3ai8 A 2.11 BS01 HNQ A 1 Q23 G24 S25 C26 H110 H111 C119 W221 Q25 G26 S27 C28 H112 H113 C121 W223 Q23 C29 H199 N219 Q25 C31 H201 N221 3.4.22.1 0006508,0008234 Ki=271.8uM Ki=271800nM P07858 21598397 255 LKLPASFDAREQWPQCPTIKEIRDQGSCGSCWAFGAVEAISDRICIHTNAHVSVEVSAEDLLTCCGSMCGDGCNGGYPAEAWNFWTRKGLVSGGLYESHVGCRPYSIPPCEHHVNGSRPPCTGEGDTPKCSKICEPGYSPTYKQDKHYGYNSYSVSNSEKDIMAEIYKNGPVEGAFSVYSDFLLYKSGVYQHVTGEMMGGHAIRILGWGVENGTPYWLVANSWNTDWGDNGFFKILRGQDHCGIESEVVAGIPRTD 3ai8 B 2.11 BS01 HNQ B 1 Q23 G24 S25 C26 H110 H111 C119 G121 W221 Q25 G26 S27 C28 H112 H113 C121 G123 W223 Q23 C29 H199 N219 Q25 C31 H201 N221 3.4.22.1 0006508,0008234 Ki=271.8uM -logKd/Ki=3.81, Ki=154.4uM Ki=271800nM P07858 21598397 255 LKLPASFDAREQWPQCPTIKEIRDQGSCGSCWAFGAVEAISDRICIHTNAHVSVEVSAEDLLTCCGSMCGDGCNGGYPAEAWNFWTRKGLVSGGLYESHVGCRPYSIPPCEHHVNGSRPPCTGEGDTPKCSKICEPGYSPTYKQDKHYGYNSYSVSNSEKDIMAEIYKNGPVEGAFSVYSDFLLYKSGVYQHVTGEMMGGHAIRILGWGVENGTPYWLVANSWNTDWGDNGFFKILRGQDHCGIESEVVAGIPRTD