2zjw A 2.4 BS01 REF A 1 L45 V53 V66 K68 F113 I174 D175 L45 V53 V66 K68 F113 I174 D175 D156 K158 N161 D175 P184 S194 D156 K158 N161 D175 P184 S194 2.7.11.1 0004672,0004674,0005524,0006468 Ki=0.02uM -logKd/Ki=7.70, Ki=0.02uM Ki=20nM, IC50=40nM P68400 19414254 336 MSGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQA