2zjf A 2.4 BS01 BSU A 1 D104 W105 I137 Y164 V193 Y272 H333 W334 D101 W102 I134 Y161 V190 Y262 H323 W324 F36 D104 W105 I127 Y164 Y272 D302 H333 F33 D101 W102 I124 Y161 Y262 D292 H323 3.3.2.10 0003824,0004301,0009636,0016787,0042803 ic50=19nM -logKd/Ki=7.72, IC50=19nM IC50=19nM P95276 18585390 360 VHRILNCRGTRIHAVADSPPDQQGPLVVLLHGFPESWYSWRHQIPALAGAGYRVVAIDQRGYGRSSKYRVQKAYRIKELVGDVVGVLDSYGAEQAFVVGHDWGAPVAWTFAWLHPDRCAGVVGISVPFAGRGVIGLPGSPFGERRPSDYHLELAGPGRVWYQDYFAVQDGIITEIEEDLRGWLLGLTYTVSGEGMMAATKAAVSMDPIDVIRAGPLCMAEGARLKDAFVYPETMPAWFTEADLDFYTGEFERSGFGGPLSFYHNIDNDWHDLADQQGKPLTPPALFIGGQYDVGTIWGAQAIERAHEVMPNYRGTHMIADVGHWIQQEAPEETNRLLLDFLGGLRP