2yiq A 1.89 BS01 YIQ A 1 L226 V234 I251 E273 M304 G307 L354 T367 D368 L16 V20 I37 E43 M74 G77 L124 T137 D138 D347 K349 N352 D368 T387 D117 K119 N122 D138 T157 2.7.11.1 0004672,0005524,0006468 ic50=12.67nM -logKd/Ki=7.90, IC50=12.67nM O96017 21907711 600 VYPKALRDEYIMSKTLGGEVKLAFERKTCKKVAIKIISKVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ