2yhd A 2.2 BS01 TES A 1 L701 L704 N705 Q711 F764 T877 M895 L31 L34 N35 Q41 F94 T207 M225 ? IC50=2.7nM, Ki=3.2nM, EC50=1.1nM P10275 21846139 1920 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ 2yhd A 2.2 BS02 AV6 A 1 K720 V730 Q733 M734 Q738 M894 I898 K50 V60 Q63 M64 Q68 M224 I228 ? Ki=23uM -logKd/Ki=4.64, Ki=23.0uM IC50=18640nM P10275 21846139 1921 PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQ