2ycr A 2.2 BS01 HCW A 1 L226 V234 K249 E273 L301 M304 E305 G307 L354 T367 D368 L16 V21 K36 E45 L73 M76 E77 G79 L126 T139 D140 D347 K349 N352 D368 T387 D119 K121 N124 D140 T159 2.7.11.1 0004672,0005524,0006468 ic50=69.6nM -logKd/Ki=7.16, IC50=69.60nM O96017 21963792 600 VYPKALRDEYIMSKTLGSGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTAKPQ