2ycq A 2.05 BS01 UPX A 1 V234 K249 E273 L303 M304 G307 L354 T367 D368 V24 K39 E48 L78 M79 G82 L129 T142 D143 D347 K349 N352 D368 T387 D122 K124 N127 D143 T162 2.7.11.1 0004672,0005524,0006468 ic50=0.14nM -logKd/Ki=9.85, IC50=0.14nM O96017 21963792 600 VYPKALRDEYIMSKTLGSGACGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ