2xh5 A 2.72 BS01 peptide C 0 E236 F238 D275 K277 E279 F310 C311 G312 T313 E315 Y316 E91 F93 D130 K132 E134 F165 C166 G167 T168 E170 Y171 D275 K277 N280 D293 T313 D130 K132 N135 D148 T168 2.7.11.1 0004672,0004674,0005524,0006468 P31751 20151677 3 ~ 12 KVTMNDFDYLKLLGKGTFGKVILVREKATGRYYAMKILRKEVIIAKDEVAHTVTESRVLQNTRHPFLTALKYAFQTHDRLCFVMEYANGGELFFHLSRERVFTEERARFYGAEIVSALEYLHSRDVVYRDIKLENLMLDKDGHIKITDFGLCKEGISDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHERLFELILMEEIRFPRTLSPEAKSLLAGLLKKDPKQRLGGGPSDAKEVMEHRFFLSINWQDVVQKKLLPPFKPQVTSEVDTRYFDDEFTAQSITQEMFEDFDYIADW 2xh5 A 2.72 BS02 X37 A 1 G161 A179 K181 M229 E230 A232 E236 T292 D293 F439 G16 A34 K36 M84 E85 A87 E91 T147 D148 F294 D275 K277 N280 D293 T313 D130 K132 N135 D148 T168 2.7.11.1 0004672,0004674,0005524,0006468 -logKd/Ki=7.57, IC50=27nM P31751 20151677 1480 KVTMNDFDYLKLLGKGTFGKVILVREKATGRYYAMKILRKEVIIAKDEVAHTVTESRVLQNTRHPFLTALKYAFQTHDRLCFVMEYANGGELFFHLSRERVFTEERARFYGAEIVSALEYLHSRDVVYRDIKLENLMLDKDGHIKITDFGLCKEGISDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHERLFELILMEEIRFPRTLSPEAKSLLAGLLKKDPKQRLGGGPSDAKEVMEHRFFLSINWQDVVQKKLLPPFKPQVTSEVDTRYFDDEFTAQSITQEMFEDFDYIADW