2xbj A 2.3 BS01 XBJ A 1 L226 A247 I286 L301 M304 G307 E308 E351 L354 L16 A36 I62 L77 M80 G83 E84 E127 L130 D347 K349 N352 D368 T387 D123 K125 N128 D144 T161 2.7.11.1 0004672,0005524,0006468 ic50=0.003uM -logKd/Ki=8.52, IC50=0.003uM IC50=30nM O96017 21186793 1513 VYPKALRDEYIMSKTLGSGAGEVKLAFERKTCKKVAIKIISKALNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILTSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQVL