2xa4 A 2.04 BS01 AZ5 A 1 L855 V863 A880 M929 Y931 L932 G935 N981 L983 G993 L13 V19 A36 M81 Y83 L84 G87 N133 L135 G145 D976 A978 R980 N981 D994 S1016 D128 A130 R132 N133 D146 S164 2.7.10.2 0004672,0004713,0005524,0006468 ic50<0.003uM -logKd/Ki=8.52, IC50=3nM IC50=58nM O60674 21138246 2131 QFEERHLKFLQQLGKFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQAHAERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM 2xa4 B 2.04 BS01 AZ5 B 1 L855 A880 M929 E930 Y931 L932 G935 N981 L983 G993 L13 A38 M76 E77 Y78 L79 G82 N128 L130 G140 D976 A978 R980 N981 D994 S1016 D123 A125 R127 N128 D141 S162 2.7.10.2 0004672,0004713,0005524,0006468 ic50<0.003uM IC50=58nM O60674 21138246 2132 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHLRDFEREIEILKSLQHDNIVKYKGVCNLKLIMEYLPYGSLRDYLQAHAERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA