2x81 A 2.91 BS01 ZZL A 1 R137 L139 G140 V147 A160 L210 Y212 A213 G216 N261 L263 A273 R11 L13 G14 V18 A31 L81 Y83 A84 G87 N132 L134 A144 D256 K258 E260 N261 T292 D127 K129 E131 N132 T146 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 -logKd/Ki=8.30, IC50=5nM IC50=34nM, Kd=6.5nM O14965 20426425 1389 QWALEDFEIGRPLGFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPLGTVYRELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIAGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSS