2x2k A 2.6 BS01 X2K A 1 L730 V738 A756 Y806 A807 G810 L881 D892 L28 V36 A54 Y104 A105 G108 L158 D169 D850 D874 A876 R878 N879 D892 D127 D151 A153 R155 N156 D169 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=6.52, IC50=0.30uM IC50=300nM P07949 20117004 2017 GPLSLSVDAFKIPKWEFPRKNLVLGKTLGEGEFGKVVKATAFHLKGRAGYTTVAVKMLKENASPSELRDLLSEFNVLKQVNHPHVIKLYGACSQDGPLLLIVEYAKYGSLRGFLRESRKVRALTMGDLISFAWQISQGMQYLAEMKLVHRDLAARNILVAEGRKMKISDFGLSRDVYEEDSYVKRSQGRIPVKWMAIESLFDHIYTTQSDVWSFGVLLWEIVTLGGNPYPGIPPERLFNLLKTGHRMERPDNCSEEMYRLMLQCWKQEPDKRPVFADISKDLEKMMVKRR