2wu7 A 2.25 BS01 V25 A 1 L162 G163 E164 V170 A184 K186 L239 E287 L290 L28 G29 E30 V36 A50 K52 L105 E153 L156 D283 K285 N288 D320 T337 D149 K151 N154 D186 T203 2.7.12.1 0004672,0005524,0006468 ic50=530nM -logKd/Ki=6.28, IC50=530nM P49761 21276940 1483 SVEDDKEGHLVCRIGDWLQERYEIVGNLGEGTFGKVVECLDHARGKSQVALKIIRNVGKYREAARLEINVLKKIKEKDKENKFLCVLMSDWFNFHGHMCIAFELLGKNTFEFLKENNFQPYPLPHVRHMAYQLCHALRFLHENQLTHTDLKPENILFVNSEFETLYNEHKSCEEKSVKNTSIRVADFGSATFDHEHHTTIVATRHYRPPEVILELGWAQPCDVWSIGCILFEYYRGFTLFQTHENREHLVMMEKILGPIPSHMIHRTRKQKYFYKGGLVWDENSSDGRYVKENCKPLKSYMLQDSLEHVQLFDLMRRMLEFDPAQRITLAEALLHPFFAGLTPEERSF