2w4i A 1.87 BS01 DGL A 1 S8 P38 Y39 G40 C70 N71 T72 T116 C181 T182 S8 P38 Y39 G40 C70 N71 T72 T116 C181 T182 D7 S8 C70 E150 C181 H183 D7 S8 C70 E150 C181 H183 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 Q9ZLT0 19097892 1256 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLKL 2w4i A 1.87 BS02 VGA B 1 P38 T41 S143 V146 P147 E150 E151 P38 T41 S143 V146 P147 E150 E151 D7 S8 C70 E150 C181 H183 D7 S8 C70 E150 C181 H183 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 -logKd/Ki=6.30, IC50=0.5uM IC50=500nM Q9ZLT0 19097892 1256 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLKL 2w4i B 1.87 BS01 DGL B 1 S8 P38 Y39 G40 C70 N71 T72 C181 T182 H183 S8 P38 Y39 G40 C70 N71 T72 C181 T182 H183 D7 S8 C70 E150 C181 H183 D7 S8 C70 E150 C181 H183 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 Q9ZLT0 19097892 1255 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLK 2w4i B 1.87 BS02 VGA B 1 P38 T41 V146 P147 E150 E151 P38 T41 V146 P147 E150 E151 D7 S8 C70 E150 C181 H183 D7 S8 C70 E150 C181 H183 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 ic50=0.5uM -logKd/Ki=6.30, IC50=0.5uM IC50=500nM Q9ZLT0 19097892 1256 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLK 2w4i E 1.87 BS01 DGL E 1 S8 P38 Y39 G40 C70 N71 T72 C181 T182 H183 S8 P38 Y39 G40 C70 N71 T72 C181 T182 H183 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 Q9ZLT0 19097892 1255 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLK 2w4i E 1.87 BS02 VGA E 1 T41 S143 V146 P147 E150 E151 T41 S143 V146 P147 E150 E151 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 ic50=0.5uM IC50=500nM Q9ZLT0 19097892 1256 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLK 2w4i F 1.87 BS01 VGA E 1 P38 V146 P147 E150 E151 P38 V146 P147 E150 E151 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 IC50=500nM Q9ZLT0 19097892 1256 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLK 2w4i F 1.87 BS02 DGL F 1 S8 P38 Y39 G40 C70 N71 T72 C181 T182 S8 P38 Y39 G40 C70 N71 T72 C181 T182 5.1.1.3 0008360,0008881,0009252,0016853,0016855,0036361,0042802,0071555 Q9ZLT0 19097892 1255 MKIGVFDSGVGGFSVLKSLLKARLFDEIIYYGDSARVPYGTKDPTTIKQFGLEALDFFKPHEIELLIVACNTASALALEEMQKYSKIPIVGVIEPSILAIKRQVEDKNAPILVLGTKATIQSNAYDNALKQQGYLNISHLATSLFVPLIEESILEGELLETCMHYYFTPLEILPEVIILGCTHFPLIAQKIEGYFMGHFALPTPPLLIHSGDAIVEYLQQKYALKNNACTFPKVEFHASGDVIWLERQAKEWLK