2w2i A 2.1 BS01 PD2 A 1 Y133 F186 H189 E191 K207 W209 K242 H277 Y121 F174 H177 E179 K195 W197 K226 H261 G171 Y178 H189 E191 H277 A289 G159 Y166 H177 E179 H261 A273 1.14.11.66 -logKd/Ki=6.04, Ki=914nM IC50=1400nM, Ki=914000nM B2RXH2 21914792 602 HTIMTFYPTMEEFADFNTYVAYMESQGAHQAGLAKVIPPKEWKARQMYDDIEDILIATPLQQVTSGQGGVFTQYHKKKKAMRVGQYRRLANSKKYQTPPHQNFADLEQRYWKSHPGNPPIYGADISGSLFEESTKQWNLGHLGTILDLLEQECGVVIEGVNTPYLYFGMWKTTFAWHTEDMDLYSINYLHFGEPKTWYVVPPEHGQHLERLARELFPDISAFLRHKVALISPTVLKENGIPFNCMTQEAGEFMVTFPYGYHAGFNHGFNCAEAINFATPRWIDYGKMAVTFSMDPFVRIVQPESY 2w2i B 2.1 BS01 PD2 B 1 Y133 F186 H189 E191 K207 W209 K242 H277 Y121 F174 H177 E179 K195 W197 K222 H257 G171 Y178 H189 E191 H277 A289 G159 Y166 H177 E179 H257 A269 1.14.11.66 IC50=1400nM, Ki=914000nM B2RXH2 21914792 402 HTIMTFYPTMEEFADFNTYVAYMESQGAHQAGLAKVIPPKEWKARQMYDDIEDILIATPLQQVTSGQGGVFTQYHKKKKAMRVGQYRRLANSKKYQTPPHQNFADLEQRYWKSHPGNPPIYGADISGSLFEESTKQWNLGHLGTILDLLEQECGVVIEGVNTPYLYFGMWKTTFAWHTEDMDLYSINYLHFGEPKTWYVVPPEHGQHLERLARELFPDLRHKVALISPTVLKENGIPFNCMTQEAGEFMVTFPYGYHAGFNHGFNCAEAINFATPRWIDYGKMAVTFSMDPFVRIVQPESYELWKH 2w2i C 2.1 BS01 PD2 C 1 Y133 F186 H189 E191 K207 W209 K242 H277 Y121 F174 H177 E179 K195 W197 K230 H265 G171 Y178 H189 E191 H277 A289 G159 Y166 H177 E179 H265 A277 1.14.11.66 IC50=1400nM, Ki=914000nM B2RXH2 21914792 502 HTIMTFYPTMEEFADFNTYVAYMESQGAHQAGLAKVIPPKEWKARQMYDDIEDILIATPLQQVTSGQGGVFTQYHKKKKAMRVGQYRRLANSKKYQTPPHQNFADLEQRYWKSHPGNPPIYGADISGSLFEESTKQWNLGHLGTILDLLEQECGVVIEGVNTPYLYFGMWKTTFAWHTEDMDLYSINYLHFGEPKTWYVVPPEHGQHLERLARELFPDISRGCEAFLRHKVALISPTVLKENGIPFNCMTQEAGEFMVTFPYGYHAGFNHGFNCAEAINFATPRWIDYGKMAVTFSMDPFVRIVQPESYELWKH