2w0x A 2.12 BS01 FE2 A 1 H199 D201 H279 H192 D194 H272 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 Q9NWT6 20822901 1350 AVASGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN 2w0x A 2.12 BS02 PD2 A 1 Y145 T196 H199 N205 F207 K214 H279 I281 N294 W296 Y138 T189 H192 N198 F200 K207 H272 I274 N287 W289 1.14.11.30,1.14.11.n4 0003714,0005112,0005515,0005634,0005654,0005737,0005829,0008198,0008270,0019826,0031406,0036139,0036140,0042803,0045663,0045746,0045892,0046872,0048471,0051059,0051213,0062101,0071532,2001214 ic50=625uM -logKd/Ki=3.20, IC50=625uM IC50=8600nM Q9NWT6 20822901 1351 AVASGSGEPREEAGALGPAWDESQLRSYSFPTRPIPRLSQSDPRAEELIENEEPVVLTDTNLVYPALKWDLEYLQENIGNGDFSVYSASTHKFLYYDEKKMANFQNFKPRSNREEMKFHEFVEKLQDIQQRGGEERLYLQQTLNDTVGRKIVMDFLGFNWNWINKQQGKRGWGQLTSNLLLIGMEGNVTPAHYDEQQNFFAQIKGYKRCILFPPDQFECLYPYPVHHPCDRQSQVDFDNPDYERFPNFQNVVGYETVVGPGDVLYIPMYWWHHIESLLNGGITITVNFWYKGAPTPKRIEYPLKAHQKVAIMRNIEKMLGEALGNPQEVGPLLNTMIKGRYN