2w08 A 1.7 BS01 CA A 1 D58 N59 E136 Q137 D138 D58 N59 E136 Q137 D138 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 205 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 A 1.7 BS02 CA A 2 E136 D138 Q148 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 206 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 A 1.7 BS03 TPO A 1 N59 Y74 E136 Q148 N59 Y74 E136 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 Kd=380uM -logKd/Ki=3.42, Kd=380uM P02743 19372378 500 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 B 1.7 BS01 CA B 1 E136 D138 Q148 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 205 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 B 1.7 BS02 CA B 2 D58 N59 E136 Q137 D138 D58 N59 E136 Q137 D138 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 206 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 B 1.7 BS03 TPO B 1 N59 Y74 E136 D138 Q148 N59 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 Kd=380uM P02743 19372378 500 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 C 1.7 BS01 CA C 1 D58 N59 E136 Q137 D138 D58 N59 E136 Q137 D138 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 205 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 C 1.7 BS02 CA C 2 E136 D138 Q148 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 206 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 C 1.7 BS03 TPO C 1 N59 Y74 E136 D138 Q148 N59 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 Kd=380uM P02743 19372378 500 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 D 1.7 BS01 CA D 1 E136 D138 Q148 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 205 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 D 1.7 BS02 CA D 2 D58 N59 E136 Q137 D138 D58 N59 E136 Q137 D138 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 206 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 D 1.7 BS03 TPO D 1 N59 Y74 E136 D138 Q148 N59 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 Kd=380uM P02743 19372378 500 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 E 1.7 BS01 CA E 1 D58 N59 E136 Q137 D138 D58 N59 E136 Q137 D138 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 205 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 E 1.7 BS02 CA E 2 E136 D138 Q148 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 P02743 19372378 206 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV 2w08 E 1.7 BS03 TPO E 1 N59 Y74 E136 D138 Q148 N59 Y74 E136 D138 Q148 ? 0001849,0002674,0005509,0005515,0005576,0005615,0005634,0006457,0006953,0030246,0042802,0044869,0044871,0045087,0045656,0046597,0046790,0046872,0048525,0051082,0051131,0061045,0062023,0070062,0072562,1903016,1903019 Kd=380uM P02743 19372378 500 HTDLSGKVFVFPRESVTDHVNLITPLEKPLQNFTLCFRAYSDLSRAYSLFSYNTQGRDNELLVYKERVGEYSLYIGRHKVTSKVIEKFPAPVHICVSWESSSGIAEFWINGTPLVKKGLRQGYFVEAQPKIVLGQEQDSYGGKFDRSQSFVGEIGDLYMWDSVLPPENILSAYQGTPLPANILDWQALNYEIRGYVIIKPLVWV