2vle	A	2.4	BS01	DZN	A	1	M124 F170 M174 W177 F292 F296 C301 C302 D457 V458 F459	M118 F164 M168 W171 F286 F290 C295 C296 D451 V452 F453	N169 K192 E268 C302 E399 E476	N163 K186 E262 C296 E393 E470	1.2.1.3	0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627			-logKd/Ki=7.10, IC50=80nM	IC50=80nM	P05091	18613661	1501 	AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS
2vle	B	2.4	BS01	DZN	B	1	M124 F170 L173 M174 W177 F292 F296 C301 D457 V458 F459	M118 F164 L167 M168 W171 F286 F290 C295 D451 V452 F453	N169 K192 E268 C302 E399 E476	N163 K186 E262 C296 E393 E470	1.2.1.3	0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627			-logKd/Ki=7.10, IC50=80nM	IC50=80nM	P05091	18613661	1501 	AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS
2vle	C	2.4	BS01	DZN	C	1	M124 F170 L173 M174 W177 F292 F296 C301 C302 D457 V458 F459	M118 F164 L167 M168 W171 F286 F290 C295 C296 D451 V452 F453	N169 K192 E268 C302 E399 E476	N163 K186 E262 C296 E393 E470	1.2.1.3	0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627				IC50=80nM	P05091	18613661	1501 	AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS
2vle	D	2.4	BS01	DZN	D	1	V120 F170 W177 F292 F296 C301 C302 C303 D457 V458 F459	V114 F164 W171 F286 F290 C295 C296 C297 D451 V452 F453	N169 K192 E268 C302 E399 E476	N163 K186 E262 C296 E393 E470	1.2.1.3	0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627				IC50=80nM	P05091	18613661	1501 	AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS
2vle	E	2.4	BS01	DZN	E	1	M124 F170 L173 M174 W177 F292 F296 C301 C302 D457 V458 F459	M118 F164 L167 M168 W171 F286 F290 C295 C296 D451 V452 F453	N169 K192 E268 C302 E399 E476	N163 K186 E262 C296 E393 E470	1.2.1.3	0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627				IC50=80nM	P05091	18613661	1501 	AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS
2vle	F	2.4	BS01	DZN	F	1	M124 F170 L173 M174 W177 F292 F296 C301 C302 D457 V458 F459	M118 F164 L167 M168 W171 F286 F290 C295 C296 D451 V452 F453	N169 K192 E268 C302 E399 E476	N163 K186 E262 C296 E393 E470	1.2.1.3	0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627				IC50=80nM	P05091	18613661	1501 	AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS
2vle	G	2.4	BS01	DZN	G	1	M124 F170 L173 M174 W177 F292 F296 C301 D457 V458 F459	M118 F164 L167 M168 W171 F286 F290 C295 D451 V452 F453	N169 K192 E268 C302 E399 E476	N163 K186 E262 C296 E393 E470	1.2.1.3	0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627				IC50=80nM	P05091	18613661	1501 	AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS
2vle	H	2.4	BS01	DZN	H	1	M124 F170 M174 W177 F292 F296 C301 C302 C303 D457 V458 F459	M118 F164 M168 W171 F286 F290 C295 C296 C297 D451 V452 F453	N169 K192 E268 C302 E399 E476	N163 K186 E262 C296 E393 E470	1.2.1.3	0004029,0004030,0005739,0005759,0005975,0006066,0006068,0008957,0009055,0016491,0016620,0018937,0046185,0051287,0070062,0106435,1903179,1905627				IC50=80nM	P05091	18613661	1501 	AVPAPNQQPEVFCNQIFINNEWHDAVSRKTFPTVNPSTGEVICQVAEGDKEDVDKAVKAARAAFQLGSPWRRMDASHRGRLLNRLADLIERDRTYLAALETLDNGKPYVISYLVDLDMVLKCLRYYAGWADKYHGKTIPIDGDFFSYTRHEPVGVCGQIIPWNFPLLMQAWKLGPALATGNVVVMKVAEQTPLTALYVANLIKEAGFPPGVVNIVPGFGPTAGAAIASHEDVDKVAFTGSTEIGRVIQVAAGSSNLKRVTLELGGKSPNIIMSDADMDWAVEQAHFALFFNQGQCCCAGSRTFVQEDIYDEFVERSVARAKSRVVGNPFDSKTEQGPQVDETQFKKILGYINTGKQEGAKLLCGGGIAADRGYFIQPTVFGDVQDGMTIAKEEIFGPVMQILKFKTIEEVVGRANNSTYGLAAAVFTKDLDKANYLSQALQAGTVWVNCYDVFGAQSPFGGYKMSGSGRELGEYGLQAYTEVKTVTVKVPQKNS