2vev A 1.8 BS01 IZ2 A 1 Y46 R47 D48 D181 F182 C215 S216 A217 I219 G220 R221 Q262 L299 Y45 R46 D47 D180 F181 C214 S215 A216 I218 G219 R220 Q261 L298 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 ic50=300nM -logKd/Ki=6.52, IC50=300nM P18031 18037290 1300 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMGDSSVQDQWKELSHEDL