2qhm A 2.0 BS01 7CS A 1 L15 V23 A36 E85 C87 E134 N135 L137 S147 L14 V18 A31 E73 C75 E122 N123 L125 S135 D130 K132 E134 N135 D148 T170 D118 K120 E122 N123 D136 T158 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=660nM -logKd/Ki=6.18, Kd=660nM O14757 17804227 500 AVPFVEDWDLVQTLGGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRPRVTS