2p59 A 2.9 BS01 peptide C 0 V55 G57 E58 V59 I61 V62 S63 R88 T89 I90 A91 P114 G116 V1 G3 E4 V5 I7 V8 S9 R34 T35 I36 A37 P60 G62 H83 D107 G163 S165 H29 D53 G109 S111 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0044423,0046718,0046872,0097264 Q91RS4 17482818 21 ~ 36 VEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTM 2p59 B 2.9 BS01 peptide C 0 T1030 Y1032 A1033 T4 Y6 A7 H1083 D1107 G1163 S1165 H57 D81 G137 S139 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0044423,0046718,0046872,0097264 Q91RS4 17482818 21 ~ 36 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2p59 B 2.9 BS02 peptide D 0 T1030 A1031 Y1032 A1033 Q1034 T1036 R1037 C1042 T1045 S1046 E1056 E1058 V1059 I1061 V1062 S1063 R1088 T1089 I1090 A1091 V1133 R1135 T4 A5 Y6 A7 Q8 T10 R11 C16 T19 S20 E30 E32 V33 I35 V36 S37 R62 T63 I64 A65 V107 R109 H1083 D1107 G1163 S1165 H57 D81 G137 S139 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0044423,0046718,0046872,0097264 Q91RS4 17482818 20 ~ 40 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS 2p59 B 2.9 BS03 GG4 B 1 Q1067 H1083 K1162 G1163 S1165 F1180 R1181 A1182 A1183 V1184 C1185 D1194 Q41 H57 K136 G137 S139 F154 R155 A156 A157 V158 C159 D168 H1083 D1107 G1163 S1165 H57 D81 G137 S139 3.6.4.13 0006508,0008233,0008236,0016020,0019062,0019087,0033644,0044423,0046718,0046872,0097264 -logKd/Ki=7.30, Ki=0.05uM Q91RS4 17482818 1208 APITAYAQQTRGLLGCIITSLTGRDKNQVEGEVQIVSTATQTFLATCINGVCWTVYHGAGTRTIASPKGPVIQMYTNVDQDLVGWPAPQGSRSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPISYLKGSSGGPLLCPAGHAVGLFRAAVCTRGVAKAVDFIPVENLETTMRS