2p2h A 1.95 BS01 994 A 1 V848 A866 K868 E885 T916 F918 C919 G922 L1035 C1045 V30 A48 K50 E67 T98 F100 C101 G104 L167 C177 D1028 A1030 R1032 N1033 D1046 D160 A162 R164 N165 D178 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=68nM -logKd/Ki=7.17, IC50=68nM IC50=68nM P35968 17253678 501 EHAERLPYDASKWEFPRDRLKLGKPLGRQVIEADAFGIDKTATCRTVAVKMLKEGATHSEHRALMSELKILIHIGHHLNVVNLLGACTKPGGPLMVITEFCKFGNLSTYLRSKRNEFVPYKVAPEDLYKDFLTLEHLICYSFQVAKGMEFLASRKCIHRDLAARNILLSEKNVVKICDFGLARLPLKWMAPETIFDRVYTIQSDVWSFGVLLWEIFSLGASPYPGVKIDEEFCRRLKEGTRMRAPDYTTPEMYQTMLDCWHGEPSQRPTFSELVEHLGNLLQANAQQDRHHH