2nru A 2.0 BS01 T12 A 1 M192 A211 K213 Y262 V263 Y264 M265 P266 N267 G268 R273 L318 M29 A48 K50 Y99 V100 Y101 M102 P103 N104 G105 R110 L155 D311 K313 A315 N316 D329 F339 T351 D148 K150 A152 N153 D166 F176 T188 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 Ki=1.2nM Q9NWZ3 17161373 600 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAMVDITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASEKFAQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 2nru B 2.0 BS01 T12 B 1 M192 A211 K213 Y262 Y264 M265 P266 N267 G268 L318 M30 A49 K51 Y100 Y102 M103 P104 N105 G106 L156 D311 K313 A315 N316 D329 F339 T351 D149 K151 A153 N154 D167 F177 T189 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 Ki=1.2nM Q9NWZ3 17161373 601 TRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAMVDITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASEKFAQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 2nru C 2.0 BS01 T12 C 1 I185 M192 V200 A211 K213 V246 Y262 M265 P266 N267 G268 R273 L318 I22 M29 V37 A48 K50 V83 Y99 M102 P103 N104 G105 R110 L155 D311 K313 A315 N316 D329 F339 T351 D148 K150 A152 N153 D166 F176 T188 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 Ki=1.2nM Q9NWZ3 17161373 602 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAMVDITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASEKFAQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT 2nru D 2.0 BS01 T12 D 1 M192 A211 K213 Y262 V263 M265 P266 N267 G268 R273 L318 M29 A48 K50 Y99 V100 M102 P103 N104 G105 R110 L155 D311 K313 A315 N316 D329 F339 T351 D148 K150 A152 N153 D166 F176 T188 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 Ki=1.2nM Q9NWZ3 17161373 603 RFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLAAMVDITTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASEKFAQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT