2jkk A 2.0 BS01 BI9 A 1 I428 A452 L501 C502 G505 N551 L553 D564 L567 I16 A40 L89 C90 G93 N139 L141 D152 L155 D546 A548 R550 N551 D564 D134 A136 R138 N139 D152 2.7.10.2 0004672,0004713,0005524,0006468 ic50=6.24nM -logKd/Ki=8.20, IC50=6.24nM Q00944 19030106 1686 RDYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNCTSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLSRLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEK