2i4z A 2.25 BS01 DRH A 1 F282 C285 Q286 S289 A292 I296 I326 M329 L330 I341 M364 H449 L453 Y473 F76 C79 Q80 S83 A86 I90 I120 M123 L124 I135 M158 H243 L247 Y267 ? 0003677,0004879,0005634,0006355 -logKd/Ki=5.70, Kd=1978nM Ki=971nM, Kd=1978nM, EC50=590nM P37231 17403688 999 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL