2hz4 A 2.8 BS01 4ST A 1 W261 Y264 L266 K294 L302 W23 Y26 L28 K56 L64 D363 A365 R367 N368 D381 P402 D125 A127 R129 N130 D143 P164 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=5.47, IC50=3425nM P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 2hz4 A 2.8 BS02 4ST C 1 Y342 F497 Q498 S500 Y104 F259 Q260 S262 D363 A365 R367 N368 D381 P402 D125 A127 R129 N130 D143 P164 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=5.47, IC50=3425nM P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 2hz4 B 2.8 BS01 4ST B 1 L248 V256 A269 K271 F317 M318 R367 L370 D381 L16 V19 A32 K34 F80 M81 R130 L133 D144 D363 A365 R367 N368 D381 P402 D126 A128 R130 N131 D144 P165 2.7.10.2 0004672,0004713,0005524,0006468 P00519 17164530 501 DKWEMERTDITMKHKLGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQ 2hz4 C 2.8 BS01 4ST A 1 F497 Q498 S500 F256 Q257 S259 D363 A365 R367 N368 D381 P402 D122 A124 R126 N127 D140 P161 2.7.10.2 0004672,0004713,0005524,0006468 P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYTVAVKTLKDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES 2hz4 C 2.8 BS02 4ST C 1 W235 Q300 W2 Q59 D363 A365 R367 N368 D381 P402 D122 A124 R126 N127 D140 P161 2.7.10.2 0004672,0004713,0005524,0006468 P00519 17164530 501 KWEMERTDITMKHKLGEVYEGVWKKYTVAVKTLKDTMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQES