2gg0 A 1.28 BS01 CO A 1 D108 H171 T202 E204 E235 D106 H169 T200 E202 E233 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H77 D95 D106 H169 R173 H176 Q180 E202 N206 Q231 E233 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0046914,0070006 P0AE18 17120228 301 ISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg0 A 1.28 BS02 CO A 2 D97 D108 E235 D95 D106 E233 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H77 D95 D106 H169 R173 H176 Q180 E202 N206 Q231 E233 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0046914,0070006 P0AE18 17120228 302 ISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE 2gg0 A 1.28 BS03 U11 A 1 Y62 H79 D97 D108 Y168 H171 F177 H178 E204 E235 Y60 H77 D95 D106 Y166 H169 F175 H176 E202 E233 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H77 D95 D106 H169 R173 H176 Q180 E202 N206 Q231 E233 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0046914,0070006 ic50=1.7uM -logKd/Ki=5.77, IC50=1.7uM IC50=1700nM P0AE18 17120228 601 ISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE