2e9v A 2.0 BS01 85A A 1 L15 A36 K38 L84 E85 Y86 C87 G90 E91 L137 D148 L14 A35 K37 L83 E84 Y85 C86 G89 E90 L136 D147 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 -logKd/Ki=7.90, Ki=12.59nM IC50=13nM O14757 1001 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL 2e9v B 2.0 BS01 85A B 1 L15 K38 L84 E85 Y86 C87 G90 E91 L137 D148 L14 K37 L83 E84 Y85 C86 G89 E90 L136 D147 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 IC50=13nM O14757 2001 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL