2e9n A 2.5 BS01 76A A 1 L15 K38 E55 L84 Y86 C87 E91 D94 L137 D148 F149 L14 K37 E54 L83 Y85 C86 E90 D93 L136 D147 F148 D130 K132 E134 N135 D148 T170 D129 K131 E133 N134 D147 T169 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=6.2nM -logKd/Ki=8.21, IC50=6.2nM EC50=>10000nM, IC50=4nM O14757 17287122 1001 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRAVDCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK