2brb A 2.1 BS01 PFQ A 1 L15 G16 V23 A36 E85 C87 L137 L14 G15 V22 A35 E81 C83 L133 D130 K132 E134 N135 D148 T170 D126 K128 E130 N131 D144 T166 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=13.7uM -logKd/Ki=4.86, Ki=13.7uM IC50=20900nM O14757 15974586 1277 AVPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKRCPENIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGAKRP