2ada A 2.4 BS01 ZN A 1 H15 H17 H214 D295 H12 H14 H211 D292 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0000255,0001666,0001701,0001829,0001889,0001890,0002314,0002467,0002636,0002686,0002901,0002906,0004000,0005737,0005764,0005829,0005886,0006154,0006157,0006196,0006915,0006939,0007155,0008270,0009117,0009168,0009897,0009986,0010460,0014074,0016020,0016787,0019239,0019722,0030217,0030324,0030890,0031410,0032261,0032263,0032264,0033077,0033089,0033632,0042100,0042110,0043066,0043084,0043605,0044209,0045580,0045582,0045987,0046059,0046061,0046085,0046101,0046103,0046111,0046632,0046638,0046872,0046936,0048286,0048541,0048566,0050728,0050850,0050852,0050862,0050870,0050900,0060169,0060205,0060407,0070161,0070242,0070244,0070254,0070256,0140928 P03958 1925539 400 TPAFNKPKVELHVHLDGAIKPETILYFGKKRGIALPADTVEELRNIIGMDKPLSLPGFLAKFDYYMPVIAGCREAIKRIAYEFVEMKAKEGVVYVEVRYSPHLLANSKVDPMPWNQTEGDVTPDDVVDLVNQGLQEGEQAFGIKVRSILCCMRHQPSWSLEVLELCKKYNQKTVVAMDLAGDETIEGSSLFPGHVEAYEGAVKNGIHRTVHAGEVGSPEVVREAVDILKTERVGHGYHTIEDEALYNRLLKENMHFEVCPWSSYLTGAWDPKTTHAVVRFKNDKANYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEEEKKELLERLYREYQ 2ada A 2.4 BS02 HPR A 1 H17 D19 F61 L62 F65 M155 A183 G184 H214 E217 D295 D296 H14 D16 F58 L59 F62 M152 A180 G181 H211 E214 D292 D293 H15 H17 H214 E217 H238 D295 H12 H14 H211 E214 H235 D292 3.5.4.4 0000255,0001666,0001701,0001829,0001889,0001890,0002314,0002467,0002636,0002686,0002901,0002906,0004000,0005737,0005764,0005829,0005886,0006154,0006157,0006196,0006915,0006939,0007155,0008270,0009117,0009168,0009897,0009986,0010460,0014074,0016020,0016787,0019239,0019722,0030217,0030324,0030890,0031410,0032261,0032263,0032264,0033077,0033089,0033632,0042100,0042110,0043066,0043084,0043605,0044209,0045580,0045582,0045987,0046059,0046061,0046085,0046101,0046103,0046111,0046632,0046638,0046872,0046936,0048286,0048541,0048566,0050728,0050850,0050852,0050862,0050870,0050900,0060169,0060205,0060407,0070161,0070242,0070244,0070254,0070256,0140928 Ki~0.1pM -logKd/Ki=13.00, Ki=0.1pM P03958 1925539 353 TPAFNKPKVELHVHLDGAIKPETILYFGKKRGIALPADTVEELRNIIGMDKPLSLPGFLAKFDYYMPVIAGCREAIKRIAYEFVEMKAKEGVVYVEVRYSPHLLANSKVDPMPWNQTEGDVTPDDVVDLVNQGLQEGEQAFGIKVRSILCCMRHQPSWSLEVLELCKKYNQKTVVAMDLAGDETIEGSSLFPGHVEAYEGAVKNGIHRTVHAGEVGSPEVVREAVDILKTERVGHGYHTIEDEALYNRLLKENMHFEVCPWSSYLTGAWDPKTTHAVVRFKNDKANYSLNTDDPLIFKSTLDTDYQMTKKDMGFTEEEFKRLNINAAKSSFLPEEEKKELLERLYREYQ