1w6j A 2.2 BS01 R71 A 1 Y98 W192 W230 H232 C233 V236 W387 F444 D455 T502 I524 W581 F696 N697 Y93 W187 W225 H227 C228 V231 W382 F439 D450 T497 I519 W576 F691 N692 G107 L156 P190 H232 S339 W387 F444 D455 T457 A458 Y503 A536 W581 Y587 F696 C700 Y704 G102 L151 P185 H227 S334 W382 F439 D450 T452 A453 Y498 A531 W576 Y582 F691 C695 Y699 5.4.99.7 0000250,0005515,0005783,0005789,0005811,0006694,0006695,0008610,0016020,0016104,0016853,0016866,0031647 -logKd/Ki=8.19, IC50=6.5nM IC50=6.5nM P48449 15525992 1733 CLRRRGGPYKTEPATDLGRWRLNCERGRQTWTYLQDERAGREQTGLEAYALGLDTKNYFKDLPKAHTAFEGALNGMTFYVGLQAEDGHWTGDYGGPLFLLPGLLITCHVARIPLPAGYREEIVRYLRSVQLPDGGWGLHIEDKSTVFGTALNYVSLRILGVGPDDPDLVRARNILHKKGGAVAIPSWGKFWLAVLNVYSWEGLNTLFPEMWLFPDWAPAHPSTLWCHCRQVYLPMSYCYAVRLSAAEDPLVQSLRQELYVEDFASIDWLAQRNNVAPDELYTPHSWLLRVVYALLNLYEHHHSAHLRQRAVQKLYEHIVADDRFTKSISIGPISKTINMLVRWYVDGPASTAFQEHVSRIPDYLWMGLDGMKMQGTNGSQIWDTAFAIQALLEAGGHHRPEFSSCLQKAHEFLRLSQVPDNPPDYQKYYRQMRKGGFSFSTLDCGWIVSDCTAEALKAVLLLQEKCPHVTEHIPRERLCDAVAVLLNMRNPDGGFATYETKRGGHLLELLNPSEVFGDIMIDYTYVECTSAVMQALKYFHKRFPEHRAAEIRETLTQGLEFCRRQQRADGSWEGSWGVCFTYGTWFGLEAFACMGQTYRDGTACAEVSRACDFLLSRQMADGGWGEDFESCEERRYLQSAQSQIHNTCWAMMGLMAVRHPDIEAQERGVRCLLEKQLPNGDWPQENIAGVFNKSCAISYTSYRNIFPIWALGRFSQLYPERALAGHP