1v0o A 1.9 BS01 INR A 1 I10 A30 K32 F79 H81 L82 D83 L132 D143 I8 A28 K30 F69 H71 L72 D73 L122 D133 D125 K127 Q129 N130 D143 K156 T163 D115 K117 Q119 N120 D133 K146 T153 2.7.11.22,2.7.11.23 0004672,0004674,0004693,0005524,0005634,0005737,0006357,0006468,0008353,0016310,0046872,0051301,0051726,0106310 ic50=5.5uM -logKd/Ki=5.26, IC50=5.50uM Q07785 14604523 2638 KYHGLEKIGEGTYGVVYKAQNNYGETFALKKIRLSTTIREISILKELKHSNIVKLYDVIHTKKRLVLVFEHLDQDLKKLLDVCEGGLESVTAKSFLLQLLNGIAYCHDRRVLHRDLKPQNLLINREGELKIADFGLARAFGIPVRKYTHEVVTLWYRAPDVLMGSKKYSTTIDIWSVGCIFAEMVNGTPLFPGVSEADQLMRIFRILGTPNSKNWPNVTELPKYDPNFTVYEPLPWESFLKGLDESGIDLLSKMLKLDPNQRITAKQALEHAYFKE 1v0o B 1.9 BS01 INR B 1 I10 A30 K32 F79 H81 L82 D83 Q84 D85 L132 D143 I8 A28 K30 F67 H69 L70 D71 Q72 D73 L120 D131 D125 K127 Q129 N130 D143 K156 T163 D113 K115 Q117 N118 D131 K144 T151 2.7.11.22,2.7.11.23 0004672,0004674,0004693,0005524,0005634,0005737,0006357,0006468,0008353,0016310,0046872,0051301,0051726,0106310 ic50=5.5uM Q07785 14604523 2638 KYHGLEKIGEGTYGVVYKAQNNYGETFALKKIRLTIREISILKELKHSNIVKLYDVIHTKKRLVLVFEHLDQDLKKLLDVCEGGLESVTAKSFLLQLLNGIAYCHDRRVLHRDLKPQNLLINREGELKIADFGLARAFGIPVRKYTHEVVTLWYRAPDVLMGSKKYSTTIDIWSVGCIFAEMVNGTPLFPGVSEADQLMRIFRILGTPNSKNWPNVTELPKYDPNFTVYEPLPWESFLKGLDESGIDLLSKMLKLDPNQRITAKQALEHAYFKE