1u0h A 2.9 BS01 MG A 1 D440 C441 D64 C65 D396 I397 D440 H516 D20 I21 D64 H140 4.6.1.1 0009190,0016849,0035556 P30803 15591060 581 MMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 1u0h A 2.9 BS02 MG A 2 D396 I397 E398 D440 D20 I21 E22 D64 D396 I397 D440 H516 D20 I21 D64 H140 4.6.1.1 0009190,0016849,0035556 P30803 15591060 582 MMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 1u0h A 2.9 BS03 FOK A 1 Y443 V506 S508 V511 T512 Y67 V130 S132 V135 T136 D396 I397 D440 H516 D20 I21 D64 H140 4.6.1.1 0009190,0016849,0035556 P30803 15591060 101 MMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 1u0h A 2.9 BS04 ONM A 1 D396 G399 F400 T401 L438 G439 D440 D20 G23 F24 T25 L62 G63 D64 D396 I397 D440 H516 D20 I21 D64 H140 4.6.1.1 0009190,0016849,0035556 -logKd/Ki=6.96, Ki=110nM P30803 15591060 100 MMFHKIYIQKHDNVSILFADIEGFTSLASQCTAQELVMTLNELFARFDKLAAENHCLRIKILGDCYYCVSGLPEARADHAHCCVEMGMDMIEAISLVREMTGVNVNMRVGIHSGRVHCGVLGLRKWQFDVWSNDVTLANHMEAGGKAGRIHITKATLSYLNGDYEVEPGCGGERNAYLKEHSIETFLIL 1u0h B 2.9 BS01 ONM A 1 D1018 N1025 D130 N137 S891 I892 S942 R1029 K1065 S13 I14 S64 R141 K177 4.6.1.1 0009190,0016849,0035556 -logKd/Ki=6.96, Ki=110nM P26769 15591060 100 HQSYDCVCVMFASIPDFKEFYTESDVNKEGLECLRLLNEIIADFDDLLSKPKFSGVEKIKTIGSTYMAATGLSAIRQYMHIGTMVEFAYALVGKLDAINKHSFNDFKLRVGINHGPVIAGVIGAQKPQYDIWGNTVNVASRMDSTGVLDKIQVTEETSLILQTLGYTCTCRGIINVKGKGDLKTYFVNT 1u0h C 2.9 BS01 MG C 1 S54 T204 D223 S16 T146 D165 E50 T55 R201 D223 Q227 E12 T17 R143 D165 Q169 ? 0003924,0005159,0005525,0005737,0005834,0005886,0007165,0007186,0007189,0007191,0007606,0010856,0016020,0016787,0019001,0031683,0031698,0031748,0031852,0035255,0046872,0051430,0071880 P04896 15591060 396 ATHRLLLLGAGESGKSTIVKQMRILHVGEKATKVQDIKNNLKEAIETIVAAMSNLVPPVELANPENQFRVDYILSVMNVPDFDFPPEFYEHAKALWEDEGVRACYERSNEYQLIDCAQYFLDKIDVIKQDDYVPSDQDLLRCRVLTSGIFETKFQVDKVNFHMFDVGGQRDERRKWIQCFNDVTAIIFVVASSSYNMVIREDNQTNRLQEALNLFKSIWNNRWLRTISVILFLNKQDLLAEKVLAGKSKIEDYFPEFARYTTPEDATPEPGEDPRVTRAKYFIRDEFLRISTASGDGRHYCYPHFTCAVDTENIRRVFNDCRDIIQRMHL 1u0h C 2.9 BS02 GSP C 1 E50 S51 G52 K53 S54 T55 D173 L198 R199 R201 T204 G225 N292 K293 D295 L296 C365 A366 V367 E12 S13 G14 K15 S16 T17 D115 L140 R141 R143 T146 G167 N234 K235 D237 L238 C307 A308 V309 E50 T55 R201 D223 Q227 E12 T17 R143 D165 Q169 ? 0003924,0005159,0005525,0005737,0005834,0005886,0007165,0007186,0007189,0007191,0007606,0010856,0016020,0016787,0019001,0031683,0031698,0031748,0031852,0035255,0046872,0051430,0071880 P04896 15591060 395 ATHRLLLLGAGESGKSTIVKQMRILHVGEKATKVQDIKNNLKEAIETIVAAMSNLVPPVELANPENQFRVDYILSVMNVPDFDFPPEFYEHAKALWEDEGVRACYERSNEYQLIDCAQYFLDKIDVIKQDDYVPSDQDLLRCRVLTSGIFETKFQVDKVNFHMFDVGGQRDERRKWIQCFNDVTAIIFVVASSSYNMVIREDNQTNRLQEALNLFKSIWNNRWLRTISVILFLNKQDLLAEKVLAGKSKIEDYFPEFARYTTPEDATPEPGEDPRVTRAKYFIRDEFLRISTASGDGRHYCYPHFTCAVDTENIRRVFNDCRDIIQRMHL