1syh A 1.8 BS01 CPW A 1 E10 Y58 P86 L87 T88 R93 L135 G138 S139 T140 L189 E190 M193 E11 Y59 P87 L88 T89 R94 L136 G139 S140 T141 L190 E191 M194 ? 0015276,0016020 Ki=393nM -logKd/Ki=6.41, Ki=393nM Ki=223nM, EC50=13900nM P19491 15591246 501 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC