1pyn A 2.2 BS01 941 A 1 Y20 R24 Y46 D48 C215 S216 A217 G220 R221 R254 G259 Q262 G283 Y19 R23 Y45 D47 C214 S215 A216 G219 R220 R253 G258 Q261 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 Ki=3.2uM -logKd/Ki=5.49, Ki=3.2uM Ki=3200nM P18031 12951078 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG