1ony A 2.15 BS01 588 A 1 Y46 D48 K120 C215 S216 A217 I219 G220 R221 Q262 T263 Q266 G283 Y45 D47 K119 C214 S215 A216 I218 G219 R220 Q261 T262 Q265 G282 D181 C215 R221 S222 Q262 D180 C214 R220 S221 Q261 3.1.3.48 0004725,0006470,0016311 -logKd/Ki=6.77, Ki=0.17uM Ki=170nM P18031 12747781 322 EMEKEFEQIDKSGSWAAIYQDIRHEASDFPCRVAKLPKNKNRNRYRDVSPFDHSRIKLHQEDNDYINASLIKMEEAQRSYILTQGPLPNTCGHFWEMVWEQKSRGVVMLNRVMEKGSLKCAQYWPQKEEKEMIFEDTNLKLTLISEDIKSYYTVRQLELENLTTQETREILHFHYTTWPDFGVPESPASFLNFLFKVRESGSLSPEHGPVVVHCSAGIGRSGTFCLADTCLLLMDKRKDPSSVDIKKVLLEMRKFRMGLIQTADQLRFSYLAVIEGAKFIMG