1nvq A 2.0 BS01 peptide B 0 E7 W9 L11 R74 Y81 E5 W7 L9 R65 Y72 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 O14757 12244092 301 ~ 305 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA 1nvq A 2.0 BS02 UCN A 1 L15 G16 V23 A36 K38 V68 E85 Y86 C87 G90 E91 E134 L137 S147 D148 L13 G14 V21 A34 K36 V59 E76 Y77 C78 G81 E82 E125 L128 S138 D139 D130 K132 E134 N135 D148 T170 D121 K123 E125 N126 D139 T161 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=5.6nM -logKd/Ki=8.25, Ki=5.6nM IC50=9.9nM, Ki=5.6nM O14757 12244092 400 VPFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMKNIKKEICINKMLNHENVVKFYGHRREGNIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLKKGA