1mqi A 1.35 BS01 FWD A 1 Y61 L90 T91 R96 L138 G141 S142 T143 L192 E193 M196 Y59 L88 T89 R94 L136 G139 S140 T141 L190 E191 M194 ? 0015276,0016020 ic50=23.53nM -logKd/Ki=7.63, IC50=23.53nM Ki=4nM, EC50=460nM P19491 12872125 401 NKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG