1me8 A 1.9 BS01 RVP A 1 M59 G316 S317 I318 C319 D358 L380 G381 R382 Y405 G407 E408 G409 M58 G195 S196 I197 C198 D237 L259 G260 R261 Y284 G286 E287 G288 1.1.1.205 0000166,0003824,0003938,0005737,0006164,0006177,0006183,0016491,0032991,0042802,0046872 Ki=65nM -logKd/Ki=7.19, Ki=65nM P50097 12235158 602 AKYYNEPCHTFNEYLLIPGLSTVDCIPSNVNLSTPLVKFQKGQQSEINLKIPLVSAIMQSVSGEKMAIALAREGGISFIFGSQSIESQAAMVHAVKNFKAHNELVDSQKRYLVGAGINTRDFRERVPALVEAGADVLCIDSSDGFSEWQKITIGWIREKYGDKVKVGAGNIVDGEGFRYLADAGADFIKIGIGGGSICITREQKGIGRGQATAVIDVVAERNKYFEETGIYIPVCSDGGIVYDYHMTLALAMGADFIMLGRYFARFEESPTRKVTINGSVMKEYWGEGSSRARNWEGVDSYVPYAGKLKDNVEASLNKVKSTMCNCGALTIPQLQSKAKITLVSSVSIVEGGAHDVI