1km3 A 1.5 BS01 UP6 A 1 D20 K72 M126 S127 P180 Q185 G202 R203 D10 K62 M116 S117 P170 Q175 G192 R193 A42 D70 K72 D75 A32 D60 K62 D65 4.1.1.23 0004590,0005829,0006207,0006221,0016831,0044205 -logKd/Ki=4.91, Ki=12.4uM Ki=12400nM O26232 11900543 2001 VMNRLILAMDLMNRDDALRVTGEVREYIDTVAIGYPLVLSEGMDIIAEFRKRFGCRIIADFKVADIPETNEKICRATFKAGADAIIVHGFPGADSVRACLNVAEEMGREVFLLTEMSHPGAEMFIQGAADEIARMGVDLGVKNYVGPSTRPERLSRLREIIGQDSFLISPGVGAQGGDPGETLRFADAIIVGRSIYLADNPAAAAAGIIESI