1fm9 A 2.1 BS01 peptide B 0 K284 L294 V298 R302 F450 E453 K58 L68 V72 R76 F224 E227 ? 0003677,0003707,0005634,0006355,0008270 P19793 10882139 630 ~ 639 NEDMPVERILEAELAVEPKTETYVEANMGLNPSSPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 1fm9 A 2.1 BS02 9CR A 1 A272 Q275 W305 F313 R316 L326 A327 V342 C432 A46 Q49 W79 F87 R90 L100 A101 V116 C206 ? 0003677,0003707,0005634,0006355,0008270 EC50=100nM, Ki=583nM, IC50=32nM, Kd=240nM P19793 10882139 201 NEDMPVERILEAELAVEPKTETYVEANMGLNPSSPNDPVTNICQAADKQLFTLVEWAKRIPHFSELPLDDQVILLRAGWNELLIASFSHRSIAVKDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMQMDKTELGCLRAIVLFNPDSKGLSNPAEVEALREKVYASLEAYCKHKYPEQPGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAP 1fm9 D 2.1 BS01 peptide E 0 E298 K301 Q314 V315 L318 K319 L468 E471 E93 K96 Q109 V110 L113 K114 L263 E266 ? 0003677,0004879,0005634,0006355 P37231 10882139 685 ~ 700 PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY 1fm9 D 2.1 BS02 570 D 1 I281 F282 G284 C285 Q286 S289 H323 Y327 L330 I341 F360 F363 M364 H449 L465 L469 Y473 I76 F77 G79 C80 Q81 S84 H118 Y122 L125 I136 F155 F158 M159 H244 L260 L264 Y268 ? 0003677,0004879,0005634,0006355 Ki=1nM -logKd/Ki=9.00, Ki=1nM Ki=1.1nM, EC50=0.338844nM, IC50=25nM P37231 10882139 200 PESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY