1ezf A 2.15 BS01 IN0 A 1 R52 F54 Y73 G180 L183 G208 L211 P292 R15 F17 Y36 G143 L146 G171 L174 P255 Y171 R218 R228 F288 Y134 R181 R191 F251 2.5.1.21 0004310,0008610,0009058,0016765,0045338,0051996 -logKd/Ki=7.25, IC50=56nM P37268 10896663 991 NSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFAKPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVKIDATNMPAVKAIIYQYMEEIYHRIPDSDPSSSKTRQIISTIRTQN 1ezf B 2.15 BS01 IN0 B 1 S51 S53 F54 Y73 L76 V179 G180 L183 L211 F288 S18 S20 F21 Y40 L43 V146 G147 L150 L178 F255 Y171 R218 R228 F288 Y138 R185 R195 F255 2.5.1.21 0004310,0008610,0009058,0016765,0045338,0051996 P37268 10896663 992 NSLSNSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFAKPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVATNMPAVKAIIYQYMEEIYHRIPDSDPSSSKTRQIISTIRTQN 1ezf C 2.15 BS01 IN0 C 1 R52 S53 F54 Y73 V179 G180 L183 M207 G208 L211 F288 R15 S16 F17 Y36 V142 G143 L146 M170 G171 L174 F251 Y171 R218 R228 F288 Y134 R181 R191 F251 2.5.1.21 0004310,0008610,0009058,0016765,0045338,0051996 P37268 10896663 995 NSLKTCYKYLNQTSRSFAAVIQALDGEMRNAVCIFYLVLRALDTLEDDMTISVEKKVPLLHNFHSFLYQPDWRFMESKEKDRQVLEDFPTISLEFRNLAEKYQTVIADICRRMGIGMAEFLDKHVTSEQEWDKYCHYVAGLVGIGLSRLFSASEFEDPLVGEDTERANSMGLFLQKTNIIRDYLEDQQGGREFWPQEVWSRYVKKLGDFAKPENIDLAVQCLNELITNALHHIPDVITYLSRLRNQSVFNFCAIPQVMAIATLAACYNNQQVFKGAVATNMPAVKAIIYQYMEEIYHRIPDSDPSSSKTRQIISTIRTQN