1eef D 1.8 BS01 GLA D 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=1.2mM P32890 11173465 104 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef E 1.8 BS01 GLA E 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=1.2mM P32890 11173465 105 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef F 1.8 BS01 GLA F 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=1.2mM P32890 11173465 106 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef G 1.8 BS01 GLA G 1 E51 Q56 Q61 W88 N90 K91 E51 Q56 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 -logKd/Ki=2.92, IC50=1.2mM P32890 11173465 107 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef G 1.8 BS02 I06 G 1 Y12 I58 Y12 I58 ? 0005576,0031640,0035821,0090729 -logKd/Ki=2.92, IC50=1.2mM P32890 11173465 108 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef H 1.8 BS01 GLA H 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 -logKd/Ki=2.92, IC50=1.2mM P32890 11173465 109 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef H 1.8 BS02 I06 H 1 Y12 I58 Y12 I58 ? 0005576,0031640,0035821,0090729 -logKd/Ki=2.92, IC50=1.2mM P32890 11173465 110 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef L 1.8 BS01 GLA L 1 E51 Q56 H57 Q61 W88 N90 K91 E51 Q56 H57 Q61 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=1.2mM P32890 11173465 111 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef L 1.8 BS02 I06 P 1 G33 K34 G33 K34 ? 0005576,0031640,0035821,0090729 P32890 11173465 117 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef M 1.8 BS01 GLA M 1 E51 Q56 H57 W88 N90 K91 E51 Q56 H57 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=1.2mM P32890 11173465 112 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef N 1.8 BS01 GLA N 1 E51 Q56 H57 W88 N90 K91 E51 Q56 H57 W88 N90 K91 ? 0005576,0031640,0035821,0090729 ic50=1.2mM P32890 11173465 113 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef O 1.8 BS01 GLA O 1 E51 Q56 W88 N90 K91 E51 Q56 W88 N90 K91 ? 0005576,0031640,0035821,0090729 P32890 11173465 114 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef O 1.8 BS02 I06 O 1 Y12 I58 Y12 I58 ? 0005576,0031640,0035821,0090729 P32890 11173465 115 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef P 1.8 BS01 I06 O 1 G33 K34 G33 K34 ? 0005576,0031640,0035821,0090729 P32890 11173465 115 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef P 1.8 BS02 GLA P 1 E51 Q56 W88 N90 K91 E51 Q56 W88 N90 K91 ? 0005576,0031640,0035821,0090729 P32890 11173465 116 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN 1eef P 1.8 BS03 I06 P 1 Y12 I58 Y12 I58 ? 0005576,0031640,0035821,0090729 P32890 11173465 117 APQTITELCSEYRNTQIYTINDKILSYTESMAGKREMVIITFKSGETFQVEVPGSQHIDSQKKAIERMKDTLRITYLTETKIDKLCVWNNKTPNSIAAISMKN