1dmt A 2.1 BS01 ZN A 1 H583 H587 E646 H530 H534 E593 H583 E584 H587 E646 D650 H711 R717 H530 E531 H534 E593 D597 H658 R664 3.4.24.11 0001786,0001822,0001890,0004175,0004222,0005515,0005737,0005769,0005802,0005886,0005903,0005925,0006508,0006518,0007611,0008021,0008233,0008237,0008238,0008270,0009986,0010814,0010815,0016020,0016485,0019233,0030163,0030324,0030424,0030425,0030667,0031410,0042277,0042447,0042803,0043025,0043627,0044306,0045121,0045202,0046449,0046872,0050435,0050769,0061837,0070012,0070062,0071345,0071492,0071493,0090399,0097242,0098793,0150094,1900273,1901612 P08473 10669592 755 GICKSSDCIKSAARLIQNMDATTEPCTDFFKYACGGWLKRNVIPETSSRYGNFDILRDELEVVLKDVLQEPKTEDIVAVQKAKALYRSCINESAIDSRGGEPLLKLLPDIYGWPVATENWEQKYGASWTAEKAIAQLNSKYGKKVLINLFVGTDDKNSVNHVIHIDQPRLGLPSRDYYECTGIYKEACTAYVDFMISVARLIRQEERLPIDENQLALEMNKVMELEKEIANATAKPEDRNDPMLLYNKMTLAQIQNNFSLEINGKPFSWLNFTNEIMSTVNISITNEEDVVVYAPEYLTKLKPILTKYSARDLQNLMSWRFIMDLVSSLSRTYKESRNAFRKALYGTTSETATWRRCANYVNGNMENAVGRLYVEAAFAGESKHVVEDLIAQIREVFIQTLDDLTWMDAETKKRAEEKALAIKERIGYPDDIVSNDNKLNNEYLELNYKEDEYFENIIQNLKFSQSKQLKKLREKVDKDEWISGAAVVNAFYSSGRNQIVFPAGILQPPFFSAQQSNSLNYGGIGMVIGHEITHGFDDNGRNFNKDGDLVDWWTQQSASNFKEQSQCMVYQYGNFSWDLAGGQHLNGINTLGENIADNGGLGQAYRAYQNYIKKNGEEKLLPGLDLNHKQLFFLNFAQVWCGTYRPEYAVNSIKTDVHSPGNFRIIGTLQNSAEFSEAFHCRKNSYMNPEKKCRVW 1dmt A 2.1 BS02 RDF A 1 R102 F106 R110 N542 A543 F544 V580 E584 H587 E646 H711 R717 R49 F53 R57 N489 A490 F491 V527 E531 H534 E593 H658 R664 H583 E584 H587 E646 D650 H711 R717 H530 E531 H534 E593 D597 H658 R664 3.4.24.11 0001786,0001822,0001890,0004175,0004222,0005515,0005737,0005769,0005802,0005886,0005903,0005925,0006508,0006518,0007611,0008021,0008233,0008237,0008238,0008270,0009986,0010814,0010815,0016020,0016485,0019233,0030163,0030324,0030424,0030425,0030667,0031410,0042277,0042447,0042803,0043025,0043627,0044306,0045121,0045202,0046449,0046872,0050435,0050769,0061837,0070012,0070062,0071345,0071492,0071493,0090399,0097242,0098793,0150094,1900273,1901612 -logKd/Ki=8.70, IC50=2nM IC50=30nM P08473 10669592 750 GICKSSDCIKSAARLIQNMDATTEPCTDFFKYACGGWLKRNVIPETSSRYGNFDILRDELEVVLKDVLQEPKTEDIVAVQKAKALYRSCINESAIDSRGGEPLLKLLPDIYGWPVATENWEQKYGASWTAEKAIAQLNSKYGKKVLINLFVGTDDKNSVNHVIHIDQPRLGLPSRDYYECTGIYKEACTAYVDFMISVARLIRQEERLPIDENQLALEMNKVMELEKEIANATAKPEDRNDPMLLYNKMTLAQIQNNFSLEINGKPFSWLNFTNEIMSTVNISITNEEDVVVYAPEYLTKLKPILTKYSARDLQNLMSWRFIMDLVSSLSRTYKESRNAFRKALYGTTSETATWRRCANYVNGNMENAVGRLYVEAAFAGESKHVVEDLIAQIREVFIQTLDDLTWMDAETKKRAEEKALAIKERIGYPDDIVSNDNKLNNEYLELNYKEDEYFENIIQNLKFSQSKQLKKLREKVDKDEWISGAAVVNAFYSSGRNQIVFPAGILQPPFFSAQQSNSLNYGGIGMVIGHEITHGFDDNGRNFNKDGDLVDWWTQQSASNFKEQSQCMVYQYGNFSWDLAGGQHLNGINTLGENIADNGGLGQAYRAYQNYIKKNGEEKLLPGLDLNHKQLFFLNFAQVWCGTYRPEYAVNSIKTDVHSPGNFRIIGTLQNSAEFSEAFHCRKNSYMNPEKKCRVW