1dls A 2.3 BS01 NDP A 1 A9 I16 G17 G20 D21 W24 G53 K54 K55 T56 S59 L75 S76 R77 E78 R91 V115 G117 S118 S119 V120 T146 A9 I16 G17 G20 D21 W24 G53 K54 K55 T56 S59 L75 S76 R77 E78 R91 V115 G117 S118 S119 V120 T146 Y22 E30 Y22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 P00374 7890613 187 VGSLNCIVAVSQNMGIGKNGDYPWPPLRNEFRYFQRMTTTSSVEGKQNLVIMGKKTWFSIPEKNRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND 1dls A 2.3 BS02 MTX A 1 I7 V8 E30 F31 F34 Q35 N64 L67 R70 I7 V8 E30 F31 F34 Q35 N64 L67 R70 Y22 E30 Y22 E30 1.5.1.3 0000900,0003723,0003729,0004146,0005542,0005737,0005739,0005829,0006729,0006730,0008144,0016491,0017148,0031103,0031427,0046452,0046653,0046654,0046655,0050661,0051000,0070402,1990825,2000121 Ki=10.9nM IC50=22nM, Kd=0.194984nM, Ki=4420nM, EC50=13.3nM P00374 7890613 188 VGSLNCIVAVSQNMGIGKNGDYPWPPLRNEFRYFQRMTTTSSVEGKQNLVIMGKKTWFSIPEKNRPLKGRINLVLSRELKEPPQGAHFLSRSLDDALKLTEQPELANKVDMVWIVGGSSVYKEAMNHPGHLKLFVTRIMQDFESDTFFPEIDLEKYKLLPEYPGVLSDVQEEKGIKYKFEVYEKND