1c3b A 2.25 BS01 BZB A 1 S64 Y150 N152 Y221 G317 A318 S61 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 -logKd/Ki=7.57, Ki=27nM IC50=200nM, Ki=27nM P00811 10595535 362 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ 1c3b B 2.25 BS01 BZB B 1 S64 Q120 Y150 N152 Y221 G317 A318 S61 Q117 Y147 N149 Y218 G314 A315 S64 K67 Y112 A114 V121 Y150 G156 E272 K315 A318 S61 K64 Y109 A111 V118 Y147 G153 E269 K312 A315 3.5.2.6 0008800,0016787,0017001,0030288,0042597,0046677 IC50=200nM, Ki=27nM P00811 10595535 362 APQQINDIVHRTITPLIEQQKIPGMAVAVIYQGKPYYFTWGYADIAKKQPVTQQTLFELGSVSKTFTGVLGGDAIARGEIKLSDPTTKYWPELTAKQWNGITLLHLATYTAGGLPLQVPDEVKSSSDLLRFYQNWQPAWAPGTQRLYANSSIGLFGALAVKPSGLSFEQAMQTRVFQPLKLNHTWINVPPAEEKNYAWGYREGKAVHVSPGALDAEAYGVKSTIEDMARWVQSNLKPLDINEKTLQQGIQLAQSRYWQTGDMYQGLGWEMLDWPVNPDSIINGSDNKIALAARPVKAITPPTPAVRASWVHKTGATGGFGSYVAFIPEKELGIVMLANKNYPNPARVDAAWQILNALQ