1aw1 A 2.7 BS01 PGA A 1 K11 H97 E169 L233 G235 G236 K10 H96 E168 L232 G234 G235 N9 K11 H97 E99 E169 G175 S214 N8 K10 H96 E98 E168 G174 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 -logKd/Ki=1.05, Ki=89mM P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAKA 1aw1 B 2.7 BS01 PGA B 1 K11 H97 E169 I174 G175 G213 S214 L233 G235 K10 H96 E168 I173 G174 G212 S213 L232 G234 N9 K11 H97 E99 E169 G175 S214 N8 K10 H96 E98 E168 G174 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 -logKd/Ki=1.05, Ki=89mM P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAK 1aw1 D 2.7 BS01 PGA D 1 K11 H97 E169 L233 G235 G236 K10 H96 E168 L232 G234 G235 N9 K11 H97 E99 E169 G175 S214 N8 K10 H96 E98 E168 G174 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAKA 1aw1 E 2.7 BS01 PGA E 1 K11 H97 E169 I174 G175 G213 S214 L233 G235 K10 H96 E168 I173 G174 G212 S213 L232 G234 N9 K11 H97 E99 E169 G175 S214 N8 K10 H96 E98 E168 G174 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAK 1aw1 G 2.7 BS01 PGA G 1 K11 H97 E169 L233 G235 G236 K10 H96 E168 L232 G234 G235 N9 K11 H97 E99 E169 G175 S214 N8 K10 H96 E98 E168 G174 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAKA 1aw1 H 2.7 BS01 PGA H 1 K11 H97 E169 I174 G175 G213 S214 L233 G235 K10 H96 E168 I173 G174 G212 S213 L232 G234 N9 K11 H97 E99 E169 G175 S214 N8 K10 H96 E98 E168 G174 S213 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAK 1aw1 J 2.7 BS01 PGA J 1 K11 H97 E169 L233 G235 G236 K10 H96 E168 L232 G234 G235 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAKA 1aw1 K 2.7 BS01 PGA K 1 K11 H97 E169 I174 G175 G213 S214 L233 G235 K10 H96 E168 I173 G174 G212 S213 L232 G234 5.3.1.1 0004807,0005737,0005829,0006094,0006096,0016853,0019563,0046166 P50921 9442062 290 RHPVVMGNWKLNGSKEMVVDLLNGLNAELEGVTGVDVAVAPPALFVDLAERTLTEAGSAIILGAQNTDLNNSGAFTGDMSPAMLKEFGATHIIIGHSERREYHAESDEFVAKKFAFLKENGLTPVLCIGESDAQNEAGETMAVCARQLDAVINTQGVEALEGAIIAYEPIWAIGTGKAATAEDAQRIHAQIRAHIAEKSEAVAKNVVIQYGGSVKPENAAAYFAQPDIDGALVGGAALDAKSFAAIAKAAAEAK