1a8t A 2.55 BS01 ZN A 1 H82 H84 H145 H82 H84 H145 H82 H84 D86 H145 C164 K167 N176 H206 H82 H84 D86 H145 C164 K167 N176 H206 3.5.2.6 0008270,0008800,0017001 P25910 9545432 251 AQKSVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIPNHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENILFGGCMLKDNQTTSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGNYGGTELIEHTKQIVNQYIESTS 1a8t A 2.55 BS02 ZN A 2 D86 H206 D86 H206 H82 H84 D86 H145 C164 K167 N176 H206 H82 H84 D86 H145 C164 K167 N176 H206 3.5.2.6 0008270,0008800,0017001 P25910 9545432 252 AQKSVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIPNHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENILFGGCMLKDNQTTSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGNYGGTELIEHTKQIVNQYIESTS 1a8t A 2.55 BS03 061 A 1 I29 W32 V35 H145 C164 D168 N176 H206 G207 I29 W32 V35 H145 C164 D168 N176 H206 G207 H82 H84 D86 H145 C164 K167 N176 H206 H82 H84 D86 H145 C164 K167 N176 H206 3.5.2.6 0008270,0008800,0017001 -logKd/Ki=5.80, Ki=1.6uM P25910 9545432 250 AQKSVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIPNHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENILFGGCMLKDNQTTSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGNYGGTELIEHTKQIVNQYIESTS 1a8t B 2.55 BS01 ZN B 1 H82 H84 H145 H80 H82 H143 H82 H84 D86 H145 C164 K167 N176 H206 H80 H82 D84 H143 C162 K165 N174 H204 3.5.2.6 0008270,0008800,0017001 P25910 9545432 251 KSVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIPNHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENILFGGCMLKDNQTTSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGNYGGTELIEHTKQIVNQYIESTS 1a8t B 2.55 BS02 ZN B 2 D86 C164 H206 D84 C162 H204 H82 H84 D86 H145 C164 K167 N176 H206 H80 H82 D84 H143 C162 K165 N174 H204 3.5.2.6 0008270,0008800,0017001 P25910 9545432 252 KSVKISDDISITQLSDKVYTYVSLAEIEGWGMVPSNGMIVINNHQAALLDTPINDAQTEMLVNWVTDSLHAKVTTFIPNHWHGDCIGGLGYLQRKGVQSYANQMTIDLAKEKGLPVPEHGFTDSLTVSLDGMPLQCYYLGGGHATDNIVVWLPTENILFGGCMLKDNQTTSIGNISDADVTAWPKTLDKVKAKFPSARYVVPGHGNYGGTELIEHTKQIVNQYIESTS