2wmx A 2.45 BS01 ZY6 A 1 V23 C87 E91 L137 V12 C66 E70 L116 D130 K132 E134 N135 D148 T170 D109 K111 E113 N114 D127 T149 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=0.86uM -logKd/Ki=6.07, IC50=0.86uM IC50=890nM O14757 19572549 1270 EDWDLVQTLGEVQLAVNRVTEEAVAVKIVDMNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPL